low affinity for EP1 and EP4 receptors and even lower affinity for EP3
a full agonist efficacy at α5 subunit (ED50=28-129 µM) and a superagonist efficacy at α4β3δ (ED50=6 µM)
A novel muscarinic receptor-independent mechanism of KCNQ2/3 potassium channel blockadeby Oxotremorine-M
Isorhamnetin 3-O-β-D-glucose-7-O-β-D-gentiobioside (30 μM) inhibits sodium oleate-induced triglyceride (TG) overloading in HepG2 cells
3'-bipyridine]-4-carboxamide
Bis-propargyl-PEG7 Catalog No.:M25097-C low affinity for EP1 andBis propargyl PEG7 is a PEG based PROTAC linker used in the synthesis of PROTACs. Bis propargyl PEG7 can be used to synthesize the polymer linked multimers of guanosine 3', 5' cyclic monophosphates. Product information CAS Number: 1351373 46 0 Molecular Weight: 402. 48 Formula: C20H34O8 Chemical Name: 4,7,10,13,16,19,22,25 octaoxaoctacosa 1,27 diyne Smiles: C#CCOCCOCCOCCOCCOCCOCCOCCOCC#C InChiKey: VVUXHSSWSXTRPE UHFFFAOYSA N InChi: InChI=1S C20H34O8